[1]
Carmena, M.; Earnshaw, W.C. The cellular geography of aurora kinases. Nat. Rev. Mol. Cell Biol., 2003, 4(11), 842-854.
[2]
Lee, E.C.; Frolov, A.; Li, R.; Ayala, G.; Greenberg, N.M. Targeting aurora kinases for the treatment of prostate cancer. Cancer Res., 2006, 66(10), 4996-5002.
[3]
Zeng, W.F.; Navaratne, K.; Prayson, R.A.; Weil, R.J. Aurora B expression correlates with aggressive behaviour in glioblastoma multiforme. J. Clin. Pathol., 2007, 60(2), 218-221.
[4]
Cheung, C.H.; Coumar, M.S.; Hsieh, H.P.; Chang, J.Y. Aurora kinase inhibitors in preclinical and clinical testing. Expert Opin. Investig. Drugs, 2009, 18(4), 379-398.
[5]
Elkins, J.M.; Santaguida, S.; Musacchio, A.; Knapp, S. Crystal structure of human aurora B in complex with INCENP and VX-680. J. Med. Chem., 2012, 55(17), 7841-7848.
[6]
Yang, J.; Ikezoe, T.; Nishioka, C.; Tasaka, T.; Taniguchi, A.; Kuwayama, Y.; Komatsu, N.; Bandobashi, K.; Togitani, K.; Koeffler, H.P.; Taguchi, H.; Yokoyama, A. AZD1152, a novel and selective Aurora B kinase inhibitor, induces growth arrest, apoptosis, and sensitization for tubulin depolymerizing agent or topoisomerase II inhibitor in human acute leukemia cells in vitro and in vivo. Blood, 2007, 110, 2034-2040.
[7]
Ju, S.; Xu, P.; Yang, X.; Sozar, S.; Muneri, C.W.; Xu, Y.; Chen, C.; Cui, P.; Xu, W.; Rui, R. Aurora B inhibitor barasertib prevents meiotic maturation and subsequent embryo development in pig oocytes. Theriogenology, 2016, 86(2), 503-515.
[8]
Tyler, R.K.; Shpiro, N.; Marquez, R.; Eyers, P.A. VX-680 inhibits aurora A and aurora B kinase activity in human cells. Cell Cyc, 2007, 6(22), 2846-2854.
[9]
Ditchfield, C.; Johnson, V.L.; Tighe, A.; Ellston, R.; Haworth, C.; Johnson, T.; Mortlock, A.; Keen, N.; Taylor, S.S. Aurora B couples chromosome alignment with anaphase by targeting BubR1, Mad2, and Cenp-E to kinetochores. J. Cell Biol., 2003, 161(2), 267-280.
[10]
Hauf, S.; Cole, R.W.; Laterra, S.; Zimmer, C.; Schnapp, G.; Walter, R.; Heckel, A.; Van Meel, J.; Rieder, C.L.; Peters, J.M. The small molecule Hesperadin reveals a role for Aurora B in correcting kinetochore-microtubule attachment and in maintaining the spindle assembly checkpoint. J. Cell Biol., 2003, 161(2), 281-294.
[11]
Determann, R.; Dreher, J.; Baumann, K.; Preu, L.; Jones, P.G.; Totzke, F.; Schächtele, C.; Kubbutat, M.H.G.; Kunick, C. 2-Anilino-4-(benzimidazol-2-yl)pyrimidines - A multikinase inhibitor scaffold with antiproliferative activity toward cancer cell lines. Eur. J. Med. Chem., 2012, 53, 254-263.
[12]
Chern; J.W.; Jagtap, A.D.; Wang, H.C.; Chen, G.S. Indolin-2-one
derivatives as protein kinase inhibitors. U.S. Patent 2013/158373,
October 24, 2013.
[13]
Gehlhaar, D.K.; Verkhivker, G.M.; Rejto, P.A.; Sherman, C.J.; Fogel, D.R.; Fogel, L.J.; Freer, S.T. molecular recognition of the inhibitor Ag-1343 by hiv-1 protease: Conformationally flexible docking by evolutionary programming. Chem. Biol., 1995, 2(5), 317-324.
[14]
Thomsen, R.; Christensen, M.H. MolDock: A new technique for high-accuracy molecular docking. J. Med. Chem., 2006, 49(11), 3315-3321.
[15]
Sessa, F.; Mapelli, M.; Ciferri, C.; Tarricone, C.; Areces, L.B.; Schneider, T.R.; Stukenberg, P.T.; Musacchio, A. Mechanism of Aurora B Activation by INCENP and Inhibition by Hesperadin. Mol. Cell, 2005, 18(3), 379-391.
[16]
Hopfinger, A.J.; Wang, S.; Tokarski, J.S.; Jin, B.; Albuquerque, M.; Madhav, P.J.; Duraiswami, C. Construction of 3D-QSAR models using the 4D-QSAR analysis formalism. J. Am. Chem. Soc., 1997, 119(43), 10509-10524.
